Optimization of Truncated Glucagon Peptides to Achieve Selective, High Potency, Full Antagonists
Bin Yang, Vasily M. Gelfanov, Diego Pérez–Tilve, Barent DuBois, Rebecca Rohlfs, Jay J. Levy, Jonathan D. Douros, Brian Finan, John P. Mayer, Richard D. DiMarchi
Abstract
action that successfully reversed glucagon-induced glucose elevation in mice.
Topics & Concepts
ChemistryPotencyGlucagonPharmacologyBiochemistryIn vitroHormoneMedicineDiabetes Treatment and ManagementNeuropeptides and Animal PhysiologyPancreatic function and diabetes