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Discovery of a potent, Highly selective, and In vivo anti-inflammatory Efficacious, P2Y6R antagonist with a novel quinoline-pyrazole scaffold

Yabiao Zhao, Bingqian Han, Zhiyi Wei, Yuanzhe Li, Yongfang Yao, Chuanjun Song, Yongtao Duan

2024European Journal of Medicinal Chemistry11 citationsDOIOpen Access PDF

Topics & Concepts

PyrazoleChemistryAntagonistIn vivoQuinolineScaffoldAnti-inflammatoryPharmacologyStereochemistryCombinatorial chemistryBiochemistryReceptorOrganic chemistryMedicineBiologyBiotechnologyBiomedical engineeringAdenosine and Purinergic SignalingSynthesis and Biological EvaluationNeuropeptides and Animal Physiology
Discovery of a potent, Highly selective, and In vivo anti-inflammatory Efficacious, P2Y6R antagonist with a novel quinoline-pyrazole scaffold | Litcius