Structural basis for NaV1.7 inhibition by pore blockers
Jiangtao Zhang, Yiqiang Shi, Zhuo Huang, Yue Li, Bei Yang, Jianke Gong, Daohua Jiang
Topics & Concepts
Helix (gastropod)ChemistryBiophysicsConformational changeNav1.5Sodium channelChannel blockerGatingProtein structureCrystallographyStereochemistryBiochemistrySodiumBiologyCalciumOrganic chemistryEcologySnailIon channel regulation and functionNeuroscience and Neuropharmacology ResearchCardiac electrophysiology and arrhythmias