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TP0586532, a non-hydroxamate LpxC inhibitor, reduces LPS release and IL-6 production both in vitro and in vivo

Kiyoko Fujita, Iichiro Takata, Ippei Yoshida, Hajime Takashima, Hiroyuki Sugiyama

2022The Journal of Antibiotics12 citationsDOIOpen Access PDF

Topics & Concepts

LipopolysaccharideIn vivoMeropenemMicrobiologyPharmacologyCiprofloxacinIn vitroLipid AChemistryBiologyAntibioticsImmunologyBiochemistryAntibiotic resistanceBiotechnologyAntibiotic Resistance in BacteriaImmune Response and InflammationAntibiotics Pharmacokinetics and Efficacy
TP0586532, a non-hydroxamate LpxC inhibitor, reduces LPS release and IL-6 production both in vitro and in vivo | Litcius