Discovery of phenylselenoether-hydantoin hybrids as ABCB1 efflux pump modulating agents with cytotoxic and antiproliferative actions in resistant T-lymphoma
Wesam Ali, Gabriella Spengler, Annamária Kincses, Márta Nové, Cecilia Battistelli, Gniewomir Latacz, Małgorzata Starek, Monika Dąbrowska, Ewelina Honkisz-Orzechowska, Annalisa Romanelli, Manuela Monica Rasile, Ewa Szymańska, Claus Jacob, Clemens Zwergel, Jadwiga Handzlik
Topics & Concepts
EffluxChemistryCancer cellMultiple drug resistanceCytotoxic T cellPharmacologyDoxorubicinCell growthP-glycoproteinATP-binding cassette transporterCancerIn vitroCancer researchBiochemistryTransporterBiologyChemotherapyGeneticsGeneAntibioticsDrug Transport and Resistance MechanismsSynthesis and Biological EvaluationMetal complexes synthesis and properties