In vitro inhibition of human UDP-glucuronosyltransferase (UGT) 1A1 by osimertinib, and prediction of in vivo drug-drug interactions
Zhe Wang, Xiaoyu Wang, Zhen Wang, Yaqin Jia, Yuyi Feng, Lili Jiang, Yangliu Xia, Jun Cao, Yong Liu
Topics & Concepts
OsimertinibGlucuronidationPharmacologyChemistryIn vivoDrugMicrosomeDrug interactionIC50In vitroReceptorEpidermal growth factor receptorBiochemistryMedicineBiologyBiotechnologyErlotinibPI3K/AKT/mTOR signaling in cancerBiochemical and Molecular ResearchChronic Lymphocytic Leukemia Research