Insights into the structure-activity relationship of pyrimidine-sulfonamide analogues for targeting BRAF V600E protein
Tarapong Srisongkram, Dheerapat Tookkane
Topics & Concepts
PyrimidineQuantitative structure–activity relationshipChemistryDocking (animal)Computational biologySulfonamideHomology modelingStereochemistryBiochemistryBiologyEnzymeMedicineNursingComputational Drug Discovery MethodsMelanoma and MAPK PathwaysSynthesis and biological activity