Proteolysis-targeting chimeras in biotherapeutics: Current trends and future applications
Qiong Li, Li Zhou, Siyuan Qin, Zhao Huang, Bowen Li, Ruolan Liu, Mei Yang, Edouard C. Nice, Huili Zhu, Canhua Huang, Canhua Huang
Topics & Concepts
ChemistryProteolysisComputational biologyUbiquitinProteasomeSmall moleculeUbiquitin ligaseProtein degradationBiochemistryBiologyEnzymeGeneProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis