Litcius/Paper detail

Fundamental aspects of DMPK optimization of targeted protein degraders

Carina Cantrill, Prasoon Chaturvedi, Caroline Rynn, Jeannine Petrig Schaffland, Isabelle Walter, Matthias Wittwer

2020Drug Discovery Today159 citationsDOI

Topics & Concepts

Drug discoveryComputational biologyBioavailabilitySmall moleculeBiochemical engineeringComputer scienceBiologyPharmacologyBioinformaticsGeneticsEngineeringProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysHistone Deacetylase Inhibitors Research