Antitumor properties of novel sesquiterpene lactone analogs as NFκB inhibitors that bind to the IKKβ ubiquitin-like domain (ULD)
Narsimha Reddy Penthala, Meenakshisundaram Balasubramaniam, Soma Shekar Dachavaram, Earl J. Morris, Poornima Bhat‐Nakshatri, Jessica Ponder, Craig T. Jordan, Harikrishna Nakshatri, Peter A. Crooks
Topics & Concepts
ChemistryParthenolideDocking (animal)IκB kinaseCell cultureCell growthCancer cellUbiquitinHEK 293 cellsIn vitroBiochemistryNF-κBApoptosisCancerBiologyReceptorMedicineNursingGeneGeneticsSesquiterpenes and Asteraceae StudiesNatural product bioactivities and synthesisNF-κB Signaling Pathways