Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity
Yue Xu, Hangsheng Yang, Yunxuan Li, Yuying Qi, Yuying Qi, Yun Hong, Binbin Cheng, Zhao‐Yang Lu, Jiaming Zhang, Chunyi Guo, Jie Fu, Jie Fu, Chun‐Hong Chen, Ning‐Ning Shi, Jianping Cai, Ke Li, Shuanghu Wang, Ruijuan Gao, Da‐Peng Dai, Da‐Peng Dai
Topics & Concepts
ChemistryStereochemistryProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchUbiquitin and proteasome pathways