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Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity

Yue Xu, Hangsheng Yang, Yunxuan Li, Yuying Qi, Yuying Qi, Yun Hong, Binbin Cheng, Zhao‐Yang Lu, Jiaming Zhang, Chunyi Guo, Jie Fu, Jie Fu, Chun‐Hong Chen, Ning‐Ning Shi, Jianping Cai, Ke Li, Shuanghu Wang, Ruijuan Gao, Da‐Peng Dai, Da‐Peng Dai

2025European Journal of Medicinal Chemistry11 citationsDOI

Topics & Concepts

ChemistryStereochemistryProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchUbiquitin and proteasome pathways
Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity | Litcius