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Evaluation of the Disconnect between Hepatocyte and Microsome Intrinsic Clearance and In Vitro In Vivo Extrapolation Performance

Beth Williamson, Stephanie Harlfinger, Dermot F. McGinnity

2020Drug Metabolism and Disposition43 citationsDOIOpen Access PDF

Topics & Concepts

In vivoHepatocyteMicrosomeIn vitroExtrapolationMicrosomaChemistryCell biologyPharmacologyBiologyBiochemistryGeneticsMathematicsMathematical analysisLiver physiology and pathologyPancreatic function and diabetesPancreatic and Hepatic Oncology Research
Evaluation of the Disconnect between Hepatocyte and Microsome Intrinsic Clearance and In Vitro In Vivo Extrapolation Performance | Litcius