Structure-based discovery of conformationally selective inhibitors of the serotonin transporter
Isha Singh, Anubha Seth, Christian B. Billesbølle, João M. Bráz, Ramona M. Rodriguiz, Kasturi Roy, Bethlehem Bekele, Veronica Craik, Xi‐Ping Huang, Danila Boytsov, Vladimir M. Pogorelov, Parnian Lak, Henry O’Donnell, Walter Sandtner, John J. Irwin, Bryan L. Roth, Allan I. Basbaum, William C. Wetsel, Aashish Manglik, Brian K. Shoichet, Gary Rudnick
Topics & Concepts
Serotonin transporterPharmacologyBiologyStereochemistrySerotoninTransporterChemistryBiochemistryReceptorGeneNeurotransmitter Receptor Influence on BehaviorReceptor Mechanisms and SignalingAnalytical Chemistry and Chromatography