Litcius/Paper detail

Structure-based discovery of conformationally selective inhibitors of the serotonin transporter

Isha Singh, Anubha Seth, Christian B. Billesbølle, João M. Bráz, Ramona M. Rodriguiz, Kasturi Roy, Bethlehem Bekele, Veronica Craik, Xi‐Ping Huang, Danila Boytsov, Vladimir M. Pogorelov, Parnian Lak, Henry O’Donnell, Walter Sandtner, John J. Irwin, Bryan L. Roth, Allan I. Basbaum, William C. Wetsel, Aashish Manglik, Brian K. Shoichet, Gary Rudnick

2023Cell94 citationsDOIOpen Access PDF

Topics & Concepts

Serotonin transporterPharmacologyBiologyStereochemistrySerotoninTransporterChemistryBiochemistryReceptorGeneNeurotransmitter Receptor Influence on BehaviorReceptor Mechanisms and SignalingAnalytical Chemistry and Chromatography