Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
Alessandro Papa, Silvia Pasquini, Francesca Galvani, Mariarosaria Cammarota, Chiara Contri, Gabriele Carullo, Sandra Gemma, Anna Ramunno, Stefania Lamponi, Beatrice Gorelli, Simona Saponara, Katia Varani, Marco Mor, Giuseppe Campiani, Francesca Boscia, Fabrizio Vincenzi, Alessio Lodola, Stefania Butini
Topics & Concepts
ChemistryMonoacylglycerol lipaseFatty acid amide hydrolaseEndocannabinoid systemNeuroprotectionPharmacologyCannabinoidCannabinoid receptorNeuroinflammationAmidaseBiochemistryAgonistEnzymeReceptorInflammationInternal medicineMedicineCannabis and Cannabinoid ResearchPharmacological Receptor Mechanisms and EffectsNeuroscience and Neuropharmacology Research