Antimicrobial evaluation of thiadiazino and thiazolo quinoxaline hybrids as potential DNA gyrase inhibitors; design, synthesis, characterization and morphological studies
Yousry A. Ammar, Awatef A. Farag, Abeer M. Ali, Sadia A. Hessein, Ahmed A. Askar, Eman A. Fayed, Doaa M. Elsisi, Ahmed Ragab
Topics & Concepts
QuinoxalineDNA gyraseChemistryAntimicrobialNorfloxacinCytotoxicityMTT assayDocking (animal)ThioureaAntibacterial activityBiochemistryIn vitroBacteriaEscherichia coliOrganic chemistryAntibioticsBiologyCiprofloxacinMedicineGeneticsGeneNursingSynthesis and Biological EvaluationSynthesis and biological activityBioactive Compounds and Antitumor Agents