Discovery of NLRP3 inhibitors using machine learning: Identification of a hit compound to treat NLRP3 activation-driven diseases
Cheng Shi, Xiangyu Zhang, Xiaowei Chi, Yi Zhou, Weiping Lyu, Tongfei Gao, Jiaxu Zhou, Yanming Chen, Chuxiao Yi, Xiaojiao Sun, Liangren Zhang, Zhenming Liu, Zhenming Liu
Topics & Concepts
In vivoChemistryDrug discoveryLead compoundPharmacologyCytotoxicitySmall moleculeIn vitroComputational biologyBiochemistryMedicineBiologyBiotechnologyInflammasome and immune disordersCholesterol and Lipid MetabolismSphingolipid Metabolism and Signaling