Litcius/Paper detail

Chalcogen- and Halogen-Bond-Donating Cyanoborohydrides Provide Imine Hydrogenation

Mikhail V. Il’in, Yana V. Safinskaya, Denis A. Polonnikov, Alexander S. Novikov, Dmitrii S. Bolotin

2024The Journal of Organic Chemistry12 citationsDOI

Abstract

Sulfonium, selenonium, telluronium, and iodonium cyanoborohydrides have been synthesized, isolated, and fully characterized by various methods, including single-crystal X-ray diffraction (XRD) analysis. The quantum theory of atoms in molecules' analysis based on the XRD data indicated that the hydride···σ-hole short contacts observed in the crystal structures of each compound have a purely noncovalent nature. The telluronium and iodonium cyanoborohydrides provide a significantly higher rate of the model reaction of imine hydrogenation compared with sodium and tetrabutylammonium cyanoborohydrides. Based on the NMR and high-resolution electrospray ionization mass spectrometry data indicating that the reaction progress is accompanied by the cation reduction, a mechanism involving intermediate formation of elusive onium hydrides has been proposed as an alternative to conventional electrophilic activation of the imine moiety by its ligation to the cation's σ-hole.

Topics & Concepts

ImineSulfoniumMoietyChemistryHalogenElectrospray ionizationElectrophileMoleculeCrystallographyMedicinal chemistryPhotochemistryPolymer chemistryOrganic chemistrySalt (chemistry)IonCatalysisAlkylCrystallography and molecular interactionsChemical Reaction MechanismsVanadium and Halogenation Chemistry