Design, synthesis and antibacterial activity of novel pleuromutilin derivatives with thieno[2,3-d]pyrimidine substitution
Rongcai Ding, Xiaoxia Wang, Jianfang Fu, Yaoyao Chang, Yingxue Li, Yajing Liu, Guoyun Liu, Jinlong Ma, Jinxing Hu
Topics & Concepts
ChemistryAntibacterial activityStaphylococcus aureusDocking (animal)PyrimidineEscherichia coliStereochemistryCytotoxicityMinimum inhibitory concentrationAntibacterial agentAntibioticsBiochemistryBacteriaIn vitroBiologyNursingGeneMedicineGeneticsVeterinary medicine and infectious diseasesSynthesis and Biological EvaluationBioactive Compounds and Antitumor Agents