Identification of aplysinopsin as a blood-brain barrier permeable scaffold for anti-cholinesterase and anti-BACE-1 activity
Vijay K. Nuthakki, Rammohan R. Yadav Bheemanaboina, Sandip B. Bharate
Topics & Concepts
ChemistryButyrylcholinesteraseAcetylcholinesteraseCholinesteraseIC50AchéEnzymeStereochemistryBlood–brain barrierIndole testPharmacologyBiochemistryBiophysicsIn vitroCombinatorial chemistryCentral nervous systemInternal medicineBiologyMedicineCholinesterase and Neurodegenerative DiseasesAlzheimer's disease research and treatmentsComputational Drug Discovery Methods