Targeting the KRAS oncogene: Synthesis, physicochemical and biological evaluation of novel G-Quadruplex DNA binders
Federica D’Aria, Vincenzo Maria D’Amore, Francesco Saverio Di Leva, Jussara Amato, Marco Caterino, Pasquale Russomanno, Silvia Salerno, Elisabetta Barresi, Marinella De Leo, Anna María Marini, Sabrina Taliani, Federico Da Settimo, Gilmar F. Salgado, Luca Pompili, Pasquale Zizza, Senji Shirasawa, Ettore Novellino, Annamaria Biroccio, Luciana Marinelli, Concetta Giancola
Topics & Concepts
KRASOncogeneG-quadruplexCancer researchChemistryColorectal cancerVirtual screeningDNASmall moleculeNucleaseBiologyComputational biologyCancerGeneBiochemistryDrug discoveryGeneticsCell cycleDNA and Nucleic Acid ChemistryAdvanced biosensing and bioanalysis techniquesRNA Interference and Gene Delivery