Evaluation of 4-aminoquinoline derivatives with an n-octylamino spacer as potential multi-targeting ligands for the treatment of Alzheimer's disease
Ana Matošević, Dejan Opsenica, Marta Spasić, Nikola Maraković, Antonio Zandona, Suzana Žunec, Marija Bartolić, Zrinka Kovarik, Anita Bosak
Topics & Concepts
TacrineButyrylcholinesteraseAcetylcholinesteraseCholinesteraseChemistryAchéPharmacologyPotencyAntioxidantEnzymeBiochemistryStereochemistryIn vitroMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments