Inverse agonism of lysophospholipids with cationic head groups at Gi-coupled receptor GPR82
Daisuke Yasuda, Fumie Hamano, Kazuyuki Masuda, Märta Dahlström, Daiki Kobayashi, Nana Sato, Takao Hamakubo, Takao Shimizu, Satoshi Ishii
Topics & Concepts
LysophosphatidylethanolamineG protein-coupled receptorInverse agonistLysophosphatidylcholineChemistryG proteinBiochemistryGi alpha subunitCell biologyReceptorAgonistPhospholipidPhosphatidylcholineBiologyMembraneReceptor Mechanisms and SignalingLipid Membrane Structure and BehaviorSphingolipid Metabolism and Signaling