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Antibody–peptide conjugates deliver covalent inhibitors blocking oncogenic cathepsins

Aaron S. Petruzzella, Marine Bruand, Albert Santamaria‐Martínez, Natalya Katanayeva, Luc Reymond, Sarah Wehrle, Sandrine Georgeon, Damla Inel, Floris J. van Dalen, David Viertl, Kelvin Lau, Florence Pojer, Margret Schottelius, Vincent Zoete, Martijn Verdoes, Caroline Arber, Bruno E. Correia, Elisa Oricchio

2024Nature Chemical Biology21 citationsDOIOpen Access PDF

Topics & Concepts

ConjugatePeptideChemistryAntibodyCovalent bondPeptidomimeticBlocking (statistics)BiochemistryBiologyImmunologyComputer scienceOrganic chemistryMathematicsComputer networkMathematical analysisMonoclonal and Polyclonal Antibodies ResearchPeptidase Inhibition and AnalysisCell Adhesion Molecules Research
Antibody–peptide conjugates deliver covalent inhibitors blocking oncogenic cathepsins | Litcius