Design, synthesis, and biological evaluation of dual-target COX-2/5-LOX inhibitors for the treatment of inflammation
Le Du, Shuaishuai Du, Jiaming Li, Hongwei Wang
Topics & Concepts
CelecoxibChemistryCyclooxygenaseArachidonate 5-lipoxygenaseZileutonPharmacologyIC50Arachidonic acidIn vivoIn vitroDocking (animal)EnzymeAnti-inflammatoryBiochemistryMedicineBiotechnologyBiologyNursingInflammatory mediators and NSAID effectsSynthesis and biological activityBioactive Compounds and Antitumor Agents