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PCSK9 inhibition with orally administered NNC0385-0434 in hypercholesterolaemia: a randomised, double-blind, placebo-controlled and active-controlled phase 2 trial

Michael J. Koren, Olivier Descamps, Yoshiki Hata, Ellen Margo Hengeveld, G. Kees Hovingh, Ignatios Ikonomidis, Maria D Radu Juul Jensen, Irene H. Langbakke, Fabrice M A C Martens, ANETTE L. SØNDERGAARD, Adam Witkowski, Wolfgang Köenig

2024The Lancet Diabetes & Endocrinology37 citationsDOIOpen Access PDF

Topics & Concepts

MedicinePCSK9PlaceboProprotein convertaseKexinSubtilisinInternal medicineOrally activeAlirocumabPharmacologyCholesterolOral administrationLipoproteinLDL receptorPathologyApolipoprotein A1ChemistryEnzymeAlternative medicineBiochemistryLipoproteins and Cardiovascular HealthCerebrovascular and Carotid Artery DiseasesPeripheral Artery Disease Management
PCSK9 inhibition with orally administered NNC0385-0434 in hypercholesterolaemia: a randomised, double-blind, placebo-controlled and active-controlled phase 2 trial | Litcius