Eco-friendly and potential colin esterase enzyme inhibitor agent sulfonyl hydrazone series: Synthesis, Bioactivity Screening, DFT, ADME properties, and Molecular Docking study
Ümmühan Özdemir Özmen, Burak Tüzün, Esra Bilen Ayan, Bekir Sıtkı Çevrimli
Topics & Concepts
ChemistryButyrylcholinesteraseAcetylcholinesteraseADMEStereochemistryCholinesteraseDocking (animal)EnzymeProtein Data Bank (RCSB PDB)Combinatorial chemistryOrganic chemistryAchéBiochemistryIn vitroPharmacologyMedicineNursingCholinesterase and Neurodegenerative DiseasesEnzyme function and inhibitionComputational Drug Discovery Methods