Bifunctional μ opioid and σ1 receptor ligands as novel analgesics with reduced side effects
Tao Zhuang, Jiaying Xiong, Shuaishuai Hao, Wei Du, Zhenming Liu, Bi‐Feng Liu, Guisen Zhang, Yin Chen
Topics & Concepts
PharmacologyOpioidChemistryμ-opioid receptorNeuropathic painChronic painAnalgesicOpioid receptorAgonistSigma-1 receptorReceptorMedicinePsychiatryBiochemistryPharmacological Receptor Mechanisms and EffectsNeuropeptides and Animal PhysiologyReceptor Mechanisms and Signaling