Synthesis, chemical characterization, PARP inhibition, DNA binding and cellular uptake of novel ruthenium(II)-arene complexes bearing benzamide derivatives in human breast cancer cells
Marijana Pavlović, Ana Tadić, Nevenka Gligorijević, Jelena M. Poljarević, Tamara Petrović, Biljana Dojčinović, Aleksandar Savić, Siniša Radulović, Sanja Grgurić‐Šipka, Sandra Aranđelović
Topics & Concepts
ChemistryPoly ADP ribose polymeraseRutheniumDNAEnzymeIn vitroBenzamideIntracellularPolymeraseCancer cellStereochemistryMolecular biologyBiochemistryCancerInternal medicineCatalysisMedicineBiologyPARP inhibition in cancer therapyMetal complexes synthesis and propertiesDNA Repair Mechanisms