Litcius/Paper detail

Inhibition of Na<sub>V</sub>1.7: the possibility of ideal analgesics

Yutaka Kitano, Tsuyoshi Shinozuka

2022RSC Medicinal Chemistry19 citationsDOIOpen Access PDF

Abstract

models and clinical results, the potential reasons behind the disconnect between preclinical results and clinical outcomes are discussed together with strategies for developing ideal analgesic agents.

Topics & Concepts

In vivoPharmacologyAnalgesicMedicineSodium channelAnalgesic agentsAdverse effectDrugChemistrySodiumBiologyOrganic chemistryBiotechnologyIon channel regulation and functionCardiac electrophysiology and arrhythmiasIon Transport and Channel Regulation