Design and synthesis of new flavonols as dual ɑ-amylase and ɑ-glucosidase inhibitors: Structure-activity relationship, drug-likeness, in vitro and in silico studies
Jamshaid Ashraf, Ehsan Ullah Mughal, Amina Sadiq, Nafeesa Naeem, Syed Aun Muhammad, Tahira Qousain, Muhammad Zafar, Bilal Ahmad Khan, M. Anees
Topics & Concepts
ChemistryIn silicoFlavonolsIn vitroDual (grammatical number)DrugDrug discoveryBiochemistryStereochemistryComputational biologyCombinatorial chemistryPharmacologyGeneQuercetinAntioxidantLiteratureArtMedicineBiologyNatural Antidiabetic Agents StudiesEnzyme Production and CharacterizationCarbohydrate Chemistry and Synthesis