Gefitinib derivatives and drug-resistance: A perspective from molecular dynamics simulations
Alireza Ahmadi, Elaheh Mohammadnejadi, Nima Razzaghi‐Asl
Topics & Concepts
GefitinibDruggabilityEpidermal growth factor receptorEGFR inhibitorsT790MChemistryMutantDocking (animal)Molecular dynamicsDrug discoveryCancer researchHydrogen bondBiologyComputational biologyBiochemistryGeneReceptorMoleculeMedicineComputational chemistryNursingOrganic chemistryLung Cancer Treatments and MutationsCancer therapeutics and mechanismsQuinazolinone synthesis and applications