Hydrophobic substrate binding pocket remodeling of echinocandin B deacylase based on multi-dimensional rational design
Heng Tang, Hanyue Zhu, Yin-feng Huang, Zeyu Wu, Shu‐Ping Zou, Zhi‐Qiang Liu, Yu‐Guo Zheng
Topics & Concepts
Rational designChemistrySubstrate (aquarium)EchinocandinStereochemistryBiologyNanotechnologyMicrobiologyAntifungalMaterials scienceEcologyFluconazolePeptidase Inhibition and AnalysisSignaling Pathways in DiseaseProtein Structure and Dynamics