Discovery of novel tranylcypromine-based derivatives as LSD1 inhibitors for gastric cancer treatment
Qisheng Ma, Yifan Zhang, Chengyang Li, Weixin Zhang, Lu Yuan, Jin-Bo Niu, Jian Song, Sai‐Yang Zhang, Hong‐Min Liu, Sai‐Yang Zhang, Hong‐Min Liu
Topics & Concepts
TranylcypromineChemistryDemethylaseEpigeneticsIC50PotencyCancer cellApoptosisPharmacologyHistone H3RegulatorCancerBiochemistryCancer researchIn vitroEnzymeInternal medicineBiologyGeneMedicineMonoamine oxidaseEpigenetics and DNA MethylationHistone Deacetylase Inhibitors ResearchCancer-related gene regulation