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Optimizing Bedaquiline for cardiotoxicity by structure based virtual screening, DFT analysis and molecular dynamic simulation studies to identify selective MDR-TB inhibitors

Iqrar Ahmad, Harsha Jadhav, Yashodeep Shinde, Vilas Jagtap, Rukaiyya T. Girase, Harun Patel

2021In Silico Pharmacology69 citationsDOIOpen Access PDF

Topics & Concepts

BedaquilinehERGVirtual screeningCardiotoxicityDocking (animal)PharmacologyChemistryDrug discoveryToxicityMedicineCombinatorial chemistryTuberculosisBiochemistryMycobacterium tuberculosisPotassium channelInternal medicinePathologyOrganic chemistryVeterinary medicineCancer therapeutics and mechanismsComputational Drug Discovery MethodsTuberculosis Research and Epidemiology
Optimizing Bedaquiline for cardiotoxicity by structure based virtual screening, DFT analysis and molecular dynamic simulation studies to identify selective MDR-TB inhibitors | Litcius