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A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 1: triazolopyrimidine, isoxazolopyrimidine and pyrrole-based (DSM) compounds

Manmohan Sharma, Vinita Pandey, Giulio Poli, Tiziano Tuccinardi, Marco L. Lolli, Vivek K. Vyas

2024Bioorganic Chemistry15 citationsDOI

Topics & Concepts

ChemistryMalariaAntimalarial AgentDrug discoveryComputational biologyPlasmodium falciparumCombinatorial chemistryBiochemistryBiologyImmunologyBiochemical and Molecular ResearchHIV/AIDS drug development and treatmentPneumocystis jirovecii pneumonia detection and treatment
A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 1: triazolopyrimidine, isoxazolopyrimidine and pyrrole-based (DSM) compounds | Litcius