Design, synthesis and evaluation of 3-amide-5-aryl benzoic acid derivatives as novel P2Y14R antagonists with potential high efficiency against acute gouty arthritis
Ran Lu, Yilin Wang, Chunxiao Liu, Zhenguo Zhang, Baiyang Li, Zibo Meng, Cheng Jiang, Qinghua Hu
Topics & Concepts
ChemistryArthritisPharmacologyBenzoic acidIn vivoAmideLead compoundInflammationBenzamideBiochemistryStereochemistryIn vitroMedicineInternal medicineBiologyBiotechnologyAdenosine and Purinergic SignalingUrticaria and Related ConditionsCardiovascular Issues in Pregnancy