Panobinostat penetrates the blood–brain barrier and achieves effective brain concentrations in a murine model
Morgan J. Homan, Andrea Franson, Karthik Ravi, Holly Roberts, Manjunath P. Pai, Cai Liu, Miao He, Aleksas Matvekas, Carl Koschmann, Bernard L. Marini
Topics & Concepts
PanobinostatPharmacokineticsCmaxPharmacologyMedicineMetaboliteChemistryInternal medicineBiochemistryHistone deacetylaseHistoneGeneHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and AnalysisAngiogenesis and VEGF in Cancer