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Review of the impact of fragment-based drug design on PROTAC degrader discovery

Peiqi Chen, Qiang Li, Xiaoguang Lei

2024TrAC Trends in Analytical Chemistry10 citationsDOI

Topics & Concepts

Drug discoveryFragment (logic)DrugComputational biologyChemistryPharmacologyComputer scienceMedicineBiologyBiochemistryAlgorithmProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments
Review of the impact of fragment-based drug design on PROTAC degrader discovery | Litcius