Litcius/Paper detail

Design, synthesis and biological evaluations of a series of Pyrido[1,2-a]pyrimidinone derivatives as novel selective FGFR inhibitors

Kai Ran, Jun Zeng, Guoquan Wan, Xiaojie He, Zhanzhan Feng, Xiang Wang, Wei Wei, Xiang Hu, Ningyu Wang, Zhihao Liu, Luoting Yu

2021European Journal of Medicinal Chemistry27 citationsDOIOpen Access PDF

Topics & Concepts

Fibroblast growth factor receptorChemistryKinaseCell growthPharmacologyCancer researchIn vitroCarcinogenesisApoptosisReceptorBiochemistryFibroblast growth factorBiologyGeneFibroblast Growth Factor ResearchKruppel-like factors researchEpigenetics and DNA Methylation
Design, synthesis and biological evaluations of a series of Pyrido[1,2-a]pyrimidinone derivatives as novel selective FGFR inhibitors | Litcius