Litcius/Paper detail

Drug repurposing and computational modeling for discovery of inhibitors of the main protease (M<sup>pro</sup>) of SARS-CoV-2

José Rogério A. Silva, Hendrik G. Kruger, Fábio Alberto de Molfetta

2021RSC Advances22 citationsDOIOpen Access PDF

Abstract

Structural and energetic features explain why some drugs can be repositioned to inhibit M pro from SARS-CoV-2.

Topics & Concepts

RepurposingDrug repositioningDrug discoverySevere acute respiratory syndrome coronavirus 2 (SARS-CoV-2)ProteaseDrugCoronavirus disease 2019 (COVID-19)ChemistryVirologyComputational biologyPharmacologyBiologyEnzymeBiochemistryMedicineEcologyInfectious disease (medical specialty)DiseasePathologyComputational Drug Discovery MethodsSARS-CoV-2 and COVID-19 Researchthermodynamics and calorimetric analyses