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Genotoxicity evaluation of ten nitrosamine drug substance-related impurities using 2D and 3D HepaRG cell models

Ji-Eun Seo, Hannah Xu, Xilin Li, Aisar Atrakchi, Timothy J. McGovern, Karen L Davis Bruno, David A. Keire, Nan Mei, Robert H. Heflich, Xiaoqing Guo

2025Regulatory Toxicology and Pharmacology8 citationsDOIOpen Access PDF

Topics & Concepts

GenotoxicityChemistryNitrosaminePharmacologyCarcinogenBiochemistryToxicityMedicineOrganic chemistryCarcinogens and Genotoxicity AssessmentSulfur Compounds in BiologyPolyamine Metabolism and Applications