Synthesis and bioevaluation of N-(3,4,5-trimethoxyphenyl)-1H-pyrazolo[3,4-b]pyridin-3-amines as tubulin polymerization inhibitors with anti-angiogenic effects
Shu-Yi Hao, Zhi-Yuan Qi, Shuai Wang, Xingrong Wang, Shi‐Wu Chen
Topics & Concepts
ChemistryTubulinStereochemistryAmine gas treatingMoietyDocking (animal)Tertiary amineMicrotubule polymerizationColchicineMicrotubuleBiochemistryCell biologyOrganic chemistryInternal medicineMedicineNursingBiologySynthesis and biological activityPhytochemical compounds biological activitiesCancer Mechanisms and Therapy