A novel class of pyrazole analogues as aurora kinase A inhibitor: design, synthesis, and anticancer evaluation
Digambar Yevale, Nishith Teraiya, Twinkle Lalwani, Rakesh Kumar Ameta, Chetan B. Sangani
Topics & Concepts
CytotoxicityChemistryApoptosisPyrazoleKinaseAurora A kinaseCell cycleVero cellAnnexinCell cycle checkpointAurora inhibitorDocking (animal)Aurora B kinaseHeLaCyclin-dependent kinase 1IC50StereochemistryBiochemistryCellIn vitroCell divisionMedicineNursingSpindle apparatusMicrotubule and mitosis dynamicsCancer-related Molecular PathwaysCancer Mechanisms and Therapy