QSAR modeling, docking, ADME and reactivity of indazole derivatives as antagonizes of estrogen receptor alpha (ER-α) positive in breast cancer
Afaf Zekri, Dalal Harkati, Samir Kenouche, Basil A. Saleh
Topics & Concepts
ChemistryADMEIndazoleQuantitative structure–activity relationshipDocking (animal)Estrogen receptorStereochemistryBreast cancerBiochemistryIn vitroMedicineInternal medicineCancerNursingComputational Drug Discovery MethodsEstrogen and related hormone effectsSynthesis and biological activity