SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease
Stefania Colarusso, Federica Ferrigno, Simona Ponzi, Francesca Pavone, Immacolata Conte, Luigi Abate, Elisa Beghetto, Antonino Missineo, Jérôme Amaudrut, Alberto Bresciani, Giacomo Paonessa, Licia Tomei, Christian Montalbetti, Elisabetta Bianchi, Carlo Toniatti, Jesus M. Ontoria
Topics & Concepts
NS3ChemistryTripeptideProteasesFlavivirusProteaseZika virusFlaviviridaeSerine proteaseBiochemistryVirologyDengue virusPeptideDengue feverVirusEnzymeBiologyHepatitis C virusMosquito-borne diseases and controlVirology and Viral DiseasesMalaria Research and Control