Litcius/Paper detail

SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease

Stefania Colarusso, Federica Ferrigno, Simona Ponzi, Francesca Pavone, Immacolata Conte, Luigi Abate, Elisa Beghetto, Antonino Missineo, Jérôme Amaudrut, Alberto Bresciani, Giacomo Paonessa, Licia Tomei, Christian Montalbetti, Elisabetta Bianchi, Carlo Toniatti, Jesus M. Ontoria

2022Bioorganic & Medicinal Chemistry11 citationsDOIOpen Access PDF

Topics & Concepts

NS3ChemistryTripeptideProteasesFlavivirusProteaseZika virusFlaviviridaeSerine proteaseBiochemistryVirologyDengue virusPeptideDengue feverVirusEnzymeBiologyHepatitis C virusMosquito-borne diseases and controlVirology and Viral DiseasesMalaria Research and Control