Inhibition of ABCG2/BCRP-mediated transport–correlation analysis of various expression systems and probe substrates
Zsolt Sáfár, Gábor Kecskeméti, Judit Molnár, Anita Kurunczi, Zoltán Szabó, Tamás Janáky, Emese Kis, Péter Krajcsi
Topics & Concepts
Abcg2ChemistrySf9IC50MembraneHEK 293 cellsPharmacologyBiophysicsATP-binding cassette transporterBiochemistryTransporterIn vitroRecombinant DNABiologyReceptorGeneSpodopteraDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesCholesterol and Lipid Metabolism