Synthesis and computational studies of new pyridine, pyrazole, pyran, and pyranopyrimidine-based derivatives of potential antimicrobial activity as DNA gyrase and topoisomerase IV inhibitors
Aisha A. Alsfouk, Ismail M. M. Othman, Manal M. Anwar, Walaa A. Alshareef, Asmaa Saleh, Eman S. Nossier
Topics & Concepts
ChemistryDNA gyraseAntimicrobialPyrazolePyridineTopoisomerasePyranCombinatorial chemistryTopoisomerase IVDNAStereochemistryBiochemistryOrganic chemistryEscherichia coliGeneSynthesis and biological activityCancer therapeutics and mechanismsSynthesis and Biological Evaluation