Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation
Emmanuel Salomon, Marjorie Schmitt, Elisabeth Mouray, Alastair G. McEwen, Lotfi Bounaadja, Morgan Torchy, Pierre Poussin‐Courmontagne, Sarah Alavi, Céline Tarnus, J. Cavarelli, Isabelle Florent, Sébastien Albrecht
Topics & Concepts
ADMEChemistryPlasmodium falciparumDrugCombinatorial chemistryLead compoundSolubilityMetabolic stabilityIC50Computational biologyPharmacologyStereochemistryBiochemistryIn vitroMalariaOrganic chemistryBiologyImmunologyMalaria Research and ControlHIV/AIDS drug development and treatmentDrug Transport and Resistance Mechanisms