Intrasubunit and Intersubunit Steroid Binding Sites Independently and Additively Mediate α1β2γ2L GABAA Receptor Potentiation by the Endogenous Neurosteroid Allopregnanolone
Allison L. Germann, Spencer R. Pierce, Hiroki Tateiwa, Yusuke Sugasawa, David E. Reichert, Alex S. Evers, Joe Henry Steinbach, Gustav Akk
Topics & Concepts
Binding siteAllosteric regulationNeuroactive steroidGABAA receptorLong-term potentiationChemistryReceptorAllopregnanoloneBiochemistryBiophysicsStereochemistryBiologyNeuroscience and Neuropharmacology ResearchReceptor Mechanisms and SignalingBioactive Compounds and Antitumor Agents