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A DNA-encoded library for the identification of natural product binders that modulate poly (ADP-ribose) polymerase 1, a validated anti-cancer target

Jie Li, Yu Li, Fengping Lu, Lili Liu, Qun Ji, Ke Song, Qianqian Yin, Richard A. Lerner, Guang Yang, Hongtao Xu, Peixiang Ma

2020Biochemical and Biophysical Research Communications17 citationsDOI

Topics & Concepts

PARP1PolymeraseNatural productLuteolinDNAPoly ADP ribose polymeraseComputational biologyDNA damageBiochemistryChemistryBiologyCombinatorial chemistryFlavonoidAntioxidantPARP inhibition in cancer therapyRNA and protein synthesis mechanismsIntegrated Circuits and Semiconductor Failure Analysis
A DNA-encoded library for the identification of natural product binders that modulate poly (ADP-ribose) polymerase 1, a validated anti-cancer target | Litcius